4byi A 2.6 BS01 FH3 A 1 R137 L139 V147 Y212 A213 P214 G216 L263 R12 L14 V22 Y87 A88 P89 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=8.05, IC50=9nM O14965 24195668 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS