4ap7 A 1.8 BS01 F47 A 1 A1108 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 F1344 A53 M105 D109 R153 M156 A166 D167 Y175 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.011uM -logKd/Ki=7.96, Ki=0.011uM Ki=11nM, IC50=7nM P08581 22924734 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF