4a6w A 1.46 BS01 MN A 1 D108 H171 E204 E235 D107 H170 E203 E234 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 0006508,0070006 22489069 1264 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 4a6w A 1.46 BS02 5C1 A 1 C59 Y62 Y65 C70 H79 D97 D108 H171 F177 H178 W221 E235 C58 Y61 Y64 C69 H78 D96 D107 H170 F176 H177 W220 E234 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 0006508,0070006 ic50=1.9uM -logKd/Ki=5.72, IC50=1.9uM 22489069 1265 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 4a6w A 1.46 BS03 MN A 2 D97 D108 E235 D96 D107 E234 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 0006508,0070006 22489069 1266 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD