3zxz A 1.8 BS01 KRW A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 D1231 F1344 I33 A53 Y104 M105 D109 R153 M156 A166 D167 Y175 D176 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.004uM -logKd/Ki=8.40, Ki=0.004uM IC50=4nM, EC50=0.300000nM, Ki=5nM P08581 22924734 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF