3uh2 A 2.0 BS01 ZN A 1 C1234 H1237 C1242 C1245 C127 H130 C135 C138 2.4.2.-,2.4.2.30 0003950 O95271 22297980 2001 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP 3uh2 A 2.0 BS02 P34 A 1 H1184 G1185 G1206 Y1213 A1215 S1221 Y1224 I1228 H80 G81 G99 Y106 A108 S114 Y117 I121 2.4.2.-,2.4.2.30 0003950 ic50=1uM -logKd/Ki=6.00, IC50=1.0uM IC50=39nM O95271 22297980 1 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP 3uh2 A 2.0 BS03 P34 A 2 F1188 I1192 F1197 D1198 H1201 F84 I88 F93 D94 H97 2.4.2.-,2.4.2.30 0003950 ic50=1uM -logKd/Ki=6.00, IC50=1.0uM IC50=39nM O95271 22297980 2 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP