3ue4 A 2.424 BS01 DB8 A 1 L248 A269 K271 V299 I313 T315 F317 M318 T319 L370 F382 L16 A37 K39 V67 I81 T83 F85 M86 T87 L138 F150 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.96, IC50=1.1nM IC50=1.1nM, Kd=0.057000nM P00519 22493660 601 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSI