3tv4 A 3.4 BS01 TV4 A 1 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 G596 A32 K34 L56 L65 I78 T80 W82 C83 F134 D145 F146 G147 D576 K578 N580 N581 D594 S616 D127 K129 N131 N132 D145 S157 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=6.96, IC50=110nM IC50=1200nM P15056 24900315 1 DDWEIPDGQITVGQRIGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK