3rvg A 2.498 BS01 17P A 1 L855 A880 E930 Y931 L932 G935 L983 L15 A40 E90 Y91 L92 G95 L143 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5nM -logKd/Ki=8.30, IC50=5nM O60674 21942426 2000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVSPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG