3ri1 A 2.1 BS01 3RH A 1 V495 A515 K517 M538 V564 A567 L633 V28 A48 K50 M71 V97 A100 L153 D626 A628 R630 N631 D644 D146 A148 R150 N151 D164 2.7.10.1 0004672,0004713,0005524,0006468 Kd=5uM -logKd/Ki=5.30, Kd=5uM IC50=1230nM P21802 21454610 2 LPEDPKWEFPRDKLTLGKPLGEGCFGQVVMAEAVGIDKDKPKEAVTVAVKMLKDDATEKDLSDLVSEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLRARRPPEQMTFKDLVSCTYQLARGMEYLASQKCIHRDLAARNVLVTENNVMKIADFGLARDINNIDYYKKTTNGRLPVKWMAPEALFDRVYTHQSDVWSFGVLMWEIFTLGGSPYPGIPVEELFKLLKEGHRMDKPANCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRILTLTT