3q96 A 3.1 BS01 0NF A 1 A481 K483 E501 L514 T529 Q530 W531 C532 H574 D594 F595 A33 K35 E53 L66 T81 Q82 W83 C84 H126 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S150 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.54, IC50=2.9nM P15056 21341678 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP