3ppj A 3.7 BS01 FOI A 1 I463 V471 A481 K483 E501 L514 I527 T529 W531 C532 F583 D594 I16 V24 A34 K36 E54 L67 I80 T82 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.70, IC50<2nM P15056 21251822 727 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK