3oy3 A 1.95 BS01 XY3 A 1 L248 A269 V270 E286 M290 V299 I315 F317 M318 I360 H361 V379 A380 D381 F382 L21 A42 V43 E59 M63 V72 I88 F90 M91 I133 H134 V152 A153 D154 F155 D363 A365 R367 N368 D381 P402 D136 A138 R140 N141 D154 P175 2.7.10.2 0004672,0004713,0005524,0006468 ic50=35.8nM -logKd/Ki=7.45, IC50=35.8nM P00520 21118377 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG