3lq8 A 2.02 BS01 88Z A 1 I1084 V1092 A1108 K1110 E1127 M1131 F1134 L1157 Y1159 M1160 G1163 H1202 M1211 A1221 D1222 F1223 I32 V40 A56 K58 E72 M76 F79 L98 Y100 M101 G104 H143 M152 A162 D163 F164 D1204 A1206 R1208 N1209 D1222 A1243 D145 A147 R149 N150 D163 A176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.4nM -logKd/Ki=9.40, IC50=0.4nM IC50=0.400000nM P08581 19808973 1 IDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRIGEVSQFLTEGIIMKDFSHPNVLSLLGICLSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDDKEYYSAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI