3kfa A 1.22 BS01 B91 A 1 L248 A269 V270 E282 E286 V289 M290 I293 I313 T315 F317 M318 G321 F359 H361 L370 A380 D381 F382 L21 A42 V43 E55 E59 V62 M63 I66 I86 T88 F90 M91 G94 F132 H134 L143 A153 D154 F155 D363 A365 R367 N368 D381 P402 D136 A138 R140 N141 D154 P175 2.7.10.2 0004672,0004713,0005524,0006468 ic50=25nM -logKd/Ki=7.60, IC50=25nM P00520 19895503 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG