3k5v A 1.74 BS01 STJ A 1 A356 L359 L360 L448 A452 E481 C483 P484 I521 L529 A113 L116 L117 L205 A209 E238 C240 P241 I278 L286 D382 A384 R386 N387 D400 P421 D139 A141 R143 N144 D157 P178 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=6.30, Kd=0.5uM P00520 20072125 1 AMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKEL 3k5v A 1.74 BS02 STI A 1 L267 Y272 A288 K290 E305 V308 M309 V318 I332 T334 F336 M337 I379 H380 L389 A399 D400 F401 L25 Y30 A46 K48 E62 V65 M66 V75 I89 T91 F93 M94 I136 H137 L146 A156 D157 F158 D382 A384 R386 N387 D400 P421 D139 A141 R143 N144 D157 P178 2.7.10.2 0004672,0004713,0005524,0006468 IC50=10.8nM P00520 20072125 2 AMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKEL