3jzi A 2.31 BS01 JZL A 1 K116 K159 A160 G164 G165 M169 Y199 E201 K202 Y203 H209 Q233 H236 L278 I287 E288 K116 K159 A160 G164 G165 M169 Y199 E201 K202 Y203 H209 Q233 H236 L278 I287 E288 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=5uM -logKd/Ki=5.30, IC50=5uM P24182 19875284 466 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG