3hq5 A 2.1 BS01 GKK A 1 L718 N719 M756 M759 L763 F778 F794 M801 L887 Y890 C891 F905 L34 N35 M72 M75 L79 F94 F109 M116 L201 Y204 C205 F219 ? ic50=16nM -logKd/Ki=7.80, IC50=16nM IC50=16nM, EC50=9nM P06401 19595590 934 QLIPPLINLLMSIEPDVIYAGHDNDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK