3g3m A 1.4 BS01 5FU A 1 S68 D70 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S35 D37 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 -logKd/Ki=5.96, Ki=1.1uM Ki=98000nM P11172 19260677 1000 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG