3g0u A 2.0 BS01 FMN A 1 A96 G97 K100 S120 N145 N181 N212 K255 N284 T285 S305 G306 V333 G334 G335 L355 Y356 T357 A61 G62 K65 S85 N110 N146 N177 K220 N249 T250 S270 G271 V298 G299 G300 L320 Y321 T322 G119 N145 F149 S215 N217 T218 K255 N284 G84 N110 F114 S180 N182 T183 K220 N249 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 19351152 398 GDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRR 3g0u A 2.0 BS02 MDY A 1 Y38 M43 P52 H56 A59 F98 R136 Y356 L359 T360 P364 Y6 M11 P20 H24 A27 F63 R101 Y321 L324 T325 P329 G119 N145 F149 S215 N217 T218 K255 N284 G84 N110 F114 S180 N182 T183 K220 N249 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 ic50=0.2uM IC50=200nM, Ki=25nM Q02127 19351152 2 GDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRR