3g0f A 2.6 BS01 B49 A 1 L595 A621 Y672 C673 C674 G676 L799 C809 F811 L30 A56 Y107 C108 C109 G111 L160 C170 F172 D792 R796 N797 D810 D153 R157 N158 D171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 -logKd/Ki=7.66, Kd=22nM Kd=0.370000nM, IC50=48nM, Ki=210nM P10721 19164557 9001 NNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFLDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARHIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISE