3fzs A 1.75 BS01 B96 A 1 E474 M478 V487 M502 L504 E509 L556 G566 D567 F568 E55 M59 V68 M83 L85 E90 L137 G147 D148 F149 D549 A551 R553 N554 D567 L587 D130 A132 R134 N135 D148 L151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.5uM -logKd/Ki=5.82, IC50=1.5uM Kd=990nM, IC50=400nM Q14289 19244237 999 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA