3fup A 2.4 BS01 MI1 A 1 L855 G856 K857 G858 G861 V863 A880 Y931 L932 L983 G993 D994 L13 G14 K15 G16 G19 V21 A38 Y85 L86 L137 G147 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=21.7nM -logKd/Ki=7.66, IC50=21.7nM IC50=77nM, EC50=93nM, Kd=5nM, Ki=0.700000nM O60674 19361440 1 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG