3fl5 A 2.3 BS01 TXQ A 1 V45 R47 V53 K68 V95 F113 V116 H160 M163 I174 D175 V39 R41 V47 K62 V89 F107 V110 H154 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0005524,0005634,0005829,0005956,0006338,0006468,0016310,0043231,0044024,0051726,0106310 -logKd/Ki=7.28, Ki=52nM P28523 19432557 338 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE