3fc2 A 2.45 BS01 IBI A 1 L59 C67 V114 E131 C133 R134 R136 F183 L23 C31 V78 E95 C97 R98 R100 F147 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=0.87nM -logKd/Ki=9.06, IC50=0.87nM IC50=0.870000nM P53350 19383823 10 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAP 3fc2 A 2.45 BS02 ZN A 1 H93 C212 H57 C176 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 P53350 19383823 8 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAP