3faa A 3.35 BS01 55F A 1 I211 A230 K232 Y249 L278 V279 S280 Y282 H283 L340 D351 I41 A60 K62 Y79 L108 V109 S110 Y112 H113 L170 D181 D333 K335 N338 D351 T375 D163 K165 N168 D181 T203 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=8.15, Ki=7.1nM Ki=7.1nM, EC50=14800nM P36897 19135364 601 ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDINHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG