3f66 A 1.4 BS01 IHX A 1 I1084 A1108 L1157 Y1159 M1160 M1211 I33 A52 L101 Y103 M104 M155 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A182 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.9uM -logKd/Ki=6.05, IC50=0.9uM IC50=900nM P08581 19059779 1 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 3f66 A 1.4 BS02 GBL A 1 M1211 A1221 D1222 Y1230 M155 A165 D166 Y174 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A182 2.7.10.1 0004672,0004713,0005524,0006468 P08581 19059779 3 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 3f66 A 1.4 BS03 GBL A 2 M1131 L1140 L1142 F1223 G1224 L1225 M75 L84 L86 F167 G168 L169 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A182 2.7.10.1 0004672,0004713,0005524,0006468 P08581 19059779 4 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 3f66 A 1.4 BS04 GBL A 3 P1176 D1180 F1216 P120 D124 F160 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A182 2.7.10.1 0004672,0004713,0005524,0006468 P08581 19059779 5 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY