3eyg A 1.9 BS01 MI1 A 1 L881 G882 E883 G884 G887 V889 A906 K908 M956 F958 L959 L1010 G1020 D1021 L17 G18 E19 G20 G23 V25 A42 K44 M84 F86 L87 L138 G148 D149 D1003 A1005 R1007 N1008 D1021 D1040 D131 A133 R135 N136 D149 D168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.6nM -logKd/Ki=8.80, IC50=1.6nM IC50=15nM, EC50=53nM, Kd=>10000nM, Ki=0.700000nM P23458 19361440 1 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK