3ewz A 1.4 BS01 CNU B 1 S257 D259 K281 H283 I368 M371 S372 I401 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 I146 M149 S150 I179 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 -logKd/Ki=4.10, IC50=79uM P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV 3ewz A 1.4 BS02 CNU B 2 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 -logKd/Ki=4.10, IC50=79uM P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV