3eou A 1.93 BS01 ZN A 1 C318 C320 C323 H349 C285 C287 C290 H316 D102 D280 C318 C320 C323 H349 D92 D253 C285 C287 C290 H316 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0016763,0046872,0101030 P28720 19894214 390 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMQSEEGVTFLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3eou A 1.93 BS02 PK3 A 1 D102 Y106 D156 C158 G229 G230 L231 A232 M260 G261 D280 D92 Y96 D129 C131 G202 G203 L204 A205 M233 G234 D253 D102 D280 C318 C320 C323 H349 D92 D253 C285 C287 C290 H316 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0016763,0046872,0101030 Ki=97nM -logKd/Ki=7.01, Ki=97nM P28720 19894214 500 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMQSEEGVTFLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF