3emg A 2.6 BS01 685 A 1 L377 F382 V385 A400 K402 M448 M450 A451 G454 L501 D512 L13 F18 V21 A35 K37 M76 M78 A79 G82 L129 D140 D494 A496 R498 N499 D512 K533 D122 A124 R126 N127 D140 K157 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.05, Ki=9nM IC50=6.0nM, Ki=9nM P43405 18938080 685 LDRKLLTLEDKELGSGNFGTVKKGYYQMKVVKTVAVKILKLKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYY