3el8 A 2.3 BS01 PD5 A 1 V281 A293 E310 M314 Y340 M341 L393 A403 D404 V24 A36 E53 M57 Y83 M84 L136 A146 D147 D386 R388 A390 N391 D404 F424 D129 R131 A133 N134 D147 F154 2.7.10.2 0004672,0004713,0005524,0006468 ic50=25nM -logKd/Ki=7.60, IC50=25nM P00523 18940662 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL