3ekn A 2.2 BS01 GS3 A 1 L1002 G1003 Q1004 V1010 A1028 V1060 M1076 M1079 G1082 M1139 L19 G20 Q21 V27 A45 V77 M93 M96 G99 M156 N1132 R1136 N1137 D1150 N149 R153 N154 D167 2.7.10.1 0004672,0004714,0005524,0006468,0007169,0016020 ic50=2nM -logKd/Ki=8.40, IC50=4nM P06213 19071018 1 YVPDEWEVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRNLAARNCMVAHDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPNMRPTFLEIVNLLKDDLHPSFPEVSFFHSEENK