3e62 A 1.922 BS01 5B1 A 1 V863 A880 M929 E930 Y931 L932 L983 V25 A42 M91 E92 Y93 L94 L145 D976 A978 R980 N981 D994 S1016 D138 A140 R142 N143 D156 S178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=40.9uM -logKd/Ki=4.39, IC50=40.9uM IC50=40900nM O60674 19019674 1 RDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA