3dkf A 1.8 BS01 SX8 A 1 I1084 A1108 L1157 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I35 A54 L103 Y105 M106 D110 R154 M157 A167 D168 Y176 D1204 A1206 R1208 N1209 D1222 D150 A152 R154 N155 D168 2.7.10.1 0004672,0004713,0005524,0006468 Ki=2.7nM -logKd/Ki=8.57, Ki=2.7nM IC50=4.0nM, Kd=0.820000nM P08581 19934279 1 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVKE