3ant A 2.4 BS01 S82 A 1 F267 D335 W336 M339 Y383 L408 Y466 H524 F36 D104 W105 M108 Y152 L177 Y235 H293 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F36 H103 D104 W105 N128 N147 Y152 Y235 D265 H293 3.1.3.76,3.3.2.10 0003824 ic50=8.5nM -logKd/Ki=8.07, IC50=8.5nM IC50=6.1nM P34913 21192659 601 CNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD