2ylq A 2.4 BS01 TES A 1 L701 L704 N705 Q711 M745 M749 F764 T877 M895 L31 L34 N35 Q41 M75 M79 F94 T207 M225 ? IC50=2.7nM, Ki=3.2nM, EC50=1.1nM P10275 22047606 1921 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ylq A 2.4 BS02 YLQ A 1 F673 N727 F826 E829 L830 N833 E837 F3 N57 F156 E159 L160 N163 E167 ? -logKd/Ki=4.30, IC50~50uM IC50=>10000nM P10275 22047606 1922 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ