2ylo A 2.5 BS01 TES A 1 L701 L704 N705 L707 M749 T877 L32 L35 N36 L38 M80 T208 ? IC50=2.7nM, Ki=3.2nM, EC50=1.1nM P10275 22047606 1920 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ylo A 2.5 BS02 YLO A 1 P723 G724 R726 N727 F826 E829 L830 N833 Y834 P54 G55 R57 N58 F157 E160 L161 N164 Y165 ? -logKd/Ki=4.88, IC50=13.1uM IC50=13100nM P10275 22047606 1922 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ