2ydk A 1.9 BS01 YDK A 1 L15 A36 E85 Y86 C87 G90 E134 N135 L137 D148 L13 A34 E78 Y79 C80 G83 E127 N128 L130 D141 D130 K132 E134 N135 D148 T170 D123 K125 E127 N128 D141 T163 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.007uM -logKd/Ki=8.15, IC50=7nM IC50=7nM, EC50=20nM O14757 22551018 1277 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK