2wtw A 3.302 BS01 ZZL A 1 R137 G140 V147 K162 L194 L210 Y212 A213 G216 L263 A273 D274 R10 G13 V20 K35 L67 L83 Y85 A86 G89 L136 A146 D147 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T159 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=8.19, Kd=6.5nM IC50=34nM, Kd=6.5nM O14965 20067443 1390 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPRGEVYKELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK