2wtv A 2.4 BS01 ZZL A 1 L139 G140 V147 K162 L194 Y212 A213 G216 L263 A273 D274 G276 V279 L15 G16 V23 K38 L70 Y88 A89 G92 L139 A149 D150 G152 V155 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki=1.8nM -logKd/Ki=8.74, Ki=1.8nM IC50=34nM, Kd=6.5nM O14965 20067443 1390 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPRGEVYKELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK