2w8y A 1.8 BS01 486 A 1 L715 L718 N719 L721 G722 E723 Q725 W755 M756 M759 F794 L797 Y890 C891 M909 L33 L36 N37 L39 G40 E41 Q43 W73 M74 M77 F112 L115 Y208 C209 M227 ? -logKd/Ki=9.09, Ki=0.82nM IC50=0.300000nM, Ki=1.1nM, EC50=>10000nM P06401 19372222 1000 LIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK