2qq7 A 2.38 BS01 SR2 A 1 A293 K295 E310 M338 M341 G344 C345 L347 D348 L393 D404 A36 K38 E42 M70 M73 G76 C77 L79 D80 L125 D136 D386 R388 A390 N391 D404 D118 R120 A122 N123 D136 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.24, IC50=5.71uM IC50=>27000nM P00523 18316192 1345 KDAWEIPRESLRLEVKLGQGFGEVWMGTWNGTTRVAIKTLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL