2qlq A 2.33 BS01 SR2 A 1 V281 A293 K295 T338 M341 C345 D348 L393 D404 V26 A38 K40 T69 M72 C76 D79 L124 D135 D386 R388 A390 N391 D404 D117 R119 A121 N122 D135 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=6.63, IC50=236nM IC50=>27000nM P00523 18316192 1345 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLAQVMKKLRHEKLVQLYAVVSEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2qlq A 2.33 BS02 SR2 A 2 C483 P484 E486 C487 E489 C195 P196 E198 C199 E201 D386 R388 A390 N391 D404 D117 R119 A121 N122 D135 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=6.63, IC50=236nM IC50=>27000nM P00523 18316192 1483 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLAQVMKKLRHEKLVQLYAVVSEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL