2q59 A 2.2 BS01 240 A 1 C285 R288 S289 A292 H323 Y327 M329 L330 L333 V339 H449 Y473 C65 R68 S69 A72 H103 Y107 M109 L110 L113 V119 H229 Y253 ? 0003677,0004879,0005634,0006355 IC50=1nM, EC50=2.0nM P37231 17937915 5001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKD