2pvk A 1.9 BS01 P45 A 1 V45 I66 K68 F113 Y115 V116 D120 H160 M163 I174 V40 I61 K63 F108 Y110 V111 D115 H155 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0005524,0005634,0005829,0005956,0006338,0006468,0016310,0043231,0044024,0051726,0106310 Ki=0.008uM -logKd/Ki=8.30, Ki=5nM P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS