2pix A 2.4 BS01 DHT A 1 L701 L704 N705 M745 M749 F764 T877 L31 L34 N35 M75 M79 F94 T207 ? IC50=>10000nM, EC50=6nM, Ki=0.2nM P10275 17911242 931 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2pix A 2.4 BS02 FLF A 1 F673 N727 E829 L830 N833 Y834 E837 F3 N57 E159 L160 N163 Y164 E167 ? -logKd/Ki=4.30, IC50=50uM IC50=>50000nM, EC50=67000nM P10275 17911242 2386 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT