2p4i A 2.5 BS01 MR9 A 1 V838 A853 E872 L879 I886 I902 Y904 A905 L971 I980 A981 D982 F983 V1 A11 E16 L23 I30 I42 Y44 A45 L111 I120 A121 D122 F123 D964 A966 R968 N969 D982 R999 D104 A106 R108 N109 D122 R134 2.7.10.1 0004672,0004713,0005524,0006468 ic50=10nM -logKd/Ki=8.00, IC50=10nM IC50=10nM Q02763 17253678 301 VLKARIRMDAAIKRGELEVLCKLGHHPNIINLLGACEHYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLSRVKKTMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGID