2ou7 A 2.4 BS01 ZN A 1 H93 C212 H57 C176 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 P53350 17461553 501 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 2ou7 A 2.4 BS02 MG A 1 E101 D194 E65 D158 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 P53350 17461553 505 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 2ou7 A 2.4 BS03 ANP A 1 G62 A80 K82 C133 F183 D194 G196 L197 G26 A44 K46 C97 F147 D158 G160 L161 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=155uM -logKd/Ki=3.81, IC50=155uM P53350 17461553 500 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA