2oiq A 2.07 BS01 STI A 1 V281 A293 I294 K295 E310 M314 I336 T338 Y340 M341 V383 H384 A403 D404 F405 V26 A38 I39 K40 E55 M59 I81 T83 Y85 M86 V128 H129 A148 D149 F150 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F156 2.7.10.2 0004672,0004713,0005524,0006468 Kd=42uM -logKd/Ki=5.00, Kd=10uM IC50=2784nM P00523 17355866 1001 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL