2jko A 1.65 BS01 BIJ A 1 R426 I428 A452 C502 T503 G505 L553 G563 D564 L567 R12 I14 A38 C88 T89 G91 L139 G149 D150 L153 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.7nM -logKd/Ki=8.11, IC50=7.7nM Q00944 19030106 1687 YEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ